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CK1-IN-1

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Catalog No. T5393Cas No. 1784751-20-7
Alias PUN51207

CK1-IN-1 (PUN51207) is a casein kinase 1 (CK1) inhibitor. CK1-IN-1 has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.

CK1-IN-1

CK1-IN-1

🥰Excellent
Purity: 98.79%
Catalog No. T5393Alias PUN51207Cas No. 1784751-20-7
CK1-IN-1 (PUN51207) is a casein kinase 1 (CK1) inhibitor. CK1-IN-1 has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.
Pack SizePriceAvailabilityQuantity
1 mg$42In Stock
2 mg$59In Stock
5 mg$98In Stock
10 mg$163In Stock
25 mg$322In Stock
50 mg$496In Stock
100 mg$745In Stock
1 mL x 10 mM (in DMSO)$108In Stock
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Purity:98.79%
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Product Introduction

Bioactivity
Description
CK1-IN-1 (PUN51207) is a casein kinase 1 (CK1) inhibitor. CK1-IN-1 has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.
Targets&IC50
CK1ε:16 nM (cell free), p38σ MAPK:73 nM (cell free), CK1δ:15 nM (cell free)
AliasPUN51207
Chemical Properties
Molecular Weight383.39
FormulaC24H15F2N3
Cas No.1784751-20-7
SmilesFc1ccc(cc1)-c1nc([nH]c1-c1ccncc1)-c1ccc2ccccc2c1F
Relative Density.1.310 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 60 mg/mL (156.5 mM)
H2O: Insoluble
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.6083 mL13.0416 mL26.0831 mL130.4155 mL
5 mM0.5217 mL2.6083 mL5.2166 mL26.0831 mL
10 mM0.2608 mL1.3042 mL2.6083 mL13.0416 mL
20 mM0.1304 mL0.6521 mL1.3042 mL6.5208 mL
50 mM0.0522 mL0.2608 mL0.5217 mL2.6083 mL
100 mM0.0261 mL0.1304 mL0.2608 mL1.3042 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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