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AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | 37 € | In Stock | |
5 mg | 93 € | In Stock | |
10 mg | 150 € | In Stock | |
25 mg | 304 € | In Stock | |
50 mg | 441 € | In Stock | |
100 mg | 615 € | In Stock | |
200 mg | 831 € | In Stock | |
1 mL x 10 mM (in DMSO) | 101 € | In Stock |
Description | AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM. |
Targets&IC50 | DYRK1B:7 nM, DYRK (pS421):0.192 μM |
In vitro | Administration of AZ-Dyrk1B-33 shows inhibition of phosphorylation of Dyrk pS421 in cells with an IC50 of 0.192 μM and no effect in sensitization[1]. |
Alias | 3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine |
Molecular Weight | 300.36 |
Formula | C19H16N4 |
Cas No. | 1679330-37-0 |
Smiles | Cc1nccc(n1)-c1cn(Cc2ccccc2)c2cnccc12 |
Relative Density. | 1.20 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 120 mg/mL (399.52 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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