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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $53 | In Stock | |
2 mg | $76 | In Stock | |
5 mg | $105 | In Stock | |
10 mg | $172 | In Stock | |
25 mg | $323 | In Stock | |
50 mg | $563 | In Stock | |
100 mg | $791 | In Stock | |
500 mg | $1,670 | In Stock |
Description | Roblitinib (FGF-401) is an inhibitor of human fibroblast growth factor receptor 4 (FGFR4), with potential antineoplastic activity. Upon administration, Roblitinib binds to and inhibits the activity of FGFR4, which leads to an inhibition of tumor cell proliferation in FGFR4-overexpressing cells. Roblitinib is a receptor tyrosine kinase upregulated in certain tumor cells and involved in tumor cell proliferation, differentiation, angiogenesis, and survival. |
In vivo | FGF-401 is a FGFR4 inhibitor developed for the treatment of solid tumor. FGF-401 is a FGFR4 inhibitor in phase I/II Clinicalal studies for the treatment of positive FGFR4 and KLB expresion solid tumors and hepatocellular carcinoma |
Alias | FGF-401 |
Molecular Weight | 506.56 |
Formula | C25H30N8O4 |
Cas No. | 1708971-55-4 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
Solubility Information | DMSO: Slightly soluble ![]() |
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