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ML254 competitively interacts with the MPEP allosteric binding site. ML254 is highly selective for mGlu5 versus other mGlu receptors, has a clean ancillary Ricerca profile, and suitable dystrophia myotonica protein kinase (DMPK) properties for systemic dosing in rodents.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | 48 € | In Stock | |
5 mg | 115 € | In Stock | |
10 mg | 187 € | In Stock | |
25 mg | 432 € | In Stock | |
50 mg | 638 € | In Stock | |
100 mg | 908 € | In Stock | |
1 mL x 10 mM (in DMSO) | 149 € | In Stock |
Description | ML254 competitively interacts with the MPEP allosteric binding site. ML254 is highly selective for mGlu5 versus other mGlu receptors, has a clean ancillary Ricerca profile, and suitable dystrophia myotonica protein kinase (DMPK) properties for systemic dosing in rodents. |
Targets&IC50 | mGluR5 (rat):8.03 nM (pEC50), mGluR5 (rat):9.3 nM (EC50) |
Molecular Weight | 310.32 |
Formula | C18H15FN2O2 |
Cas No. | 1428630-86-7 |
Smiles | CC1(COC1)NC(=O)c1ccc(cn1)C#Cc1cccc(F)c1 |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
Solubility Information | DMSO: 27.5 mg/mL (88.62 mM) | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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