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Raf inhibitor 2
🥰Excellent
Catalog No. T4194Cas No. 220904-99-4
Alias CID-25014542, CID25014542, CID 25014542
Raf inhibitor 2 (CID 25014542) is novel inhibitor of Raf kinases.
Raf inhibitor 2
🥰Excellent
Purity: 98.53%
Catalog No. T4194Alias CID-25014542, CID25014542, CID 25014542Cas No. 220904-99-4
Raf inhibitor 2 (CID 25014542) is novel inhibitor of Raf kinases.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $34 | In Stock | |
| 5 mg | $56 | In Stock | |
| 10 mg | $88 | In Stock | |
| 25 mg | $167 | In Stock | |
| 50 mg | $253 | In Stock | |
| 100 mg | $368 | In Stock | |
| 200 mg | $517 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $58 | In Stock |
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View MoreInhibitors Related to "Raf inhibitor 2"
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Sorafenib (Bay 43-9006) is a multikinase inhibitor that targets Raf-1, B-Raf, VEGFR2, VEGFR3, VEGFR4, PDGFRβ, FLT3, c-Kit, and others (IC50=6/22/90/15/20/20/57/58 nM) with oral activity. It exhibits antitumor properties and can induce autophagy, apoptosis, and agonistic iron death.
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CitedRegorafenib Cited
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CitedDabrafenib Cited
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Dabrafenib (GSK2118436A) is a Raf inhibitor that inhibits C-Raf and B-RafV600E (IC50=5/0.6 nM) and is ATP-competitive. Dabrafenib exhibits antitumor activity for the treatment of B-RafV600E-mutated melanoma.
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- $30
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Sorafenib tosylate Cited
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Sorafenib tosylate (Bay 43-9006) is a potent multikinase inhibitor (IC50s: 6/20/22 nM for Raf-1/VEGFR-3/B-Raf).
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Doramapimod
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LY3009120
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Purity:98.53%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Raf inhibitor 2 (CID 25014542) is novel inhibitor of Raf kinases. |
| Alias | CID-25014542, CID25014542, CID 25014542 |
| Molecular Weight | 429.49 |
| Formula | C15H8Br2ClNO2 |
| Cas No. | 220904-99-4 |
| Smiles | Oc1c(Br)cc(\C=C2/C(=O)Nc3ccc(Cl)cc23)cc1Br |
| Relative Density. | 1.938 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 30 mg/mL (69.85 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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