Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Sigma-1 receptor antagonist 2 is a more potent and selective antagonist of sigma 1 receptor (σ1 R, Ki = 3.88 nM) than σ2 receptor (Ki = 1288 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 97.00 | |
5 mg | In stock | $ 247.00 | |
10 mg | In stock | $ 413.00 | |
25 mg | In stock | $ 692.00 | |
50 mg | In stock | $ 985.00 | |
100 mg | In stock | $ 1,330.00 | |
500 mg | In stock | $ 2,660.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 272.00 |
Description | Sigma-1 receptor antagonist 2 is a more potent and selective antagonist of sigma 1 receptor (σ1 R, Ki = 3.88 nM) than σ2 receptor (Ki = 1288 nM). |
Targets&IC50 | σ2 receptor:1288 nM(Ki), σ1 receptor:3.88 nM(Ki) |
Molecular Weight | 375.89 |
Formula | C20H26ClN3O2 |
CAS No. | 1639220-15-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 86.67 mg/mL (230.57 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
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Sigma-1 receptor antagonist 2 1639220-15-7 GPCR/G Protein Sigma receptor σ-1 receptor antagonist 2 Sigma1 receptor antagonist 2 Sigma 1 receptor antagonist 2 Sigma Receptor Inhibitor inhibit inhibitor