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WDR5-0103

Catalog No. T3201 CAS 890190-22-4

Synonyms: WDR50103, Inhibitor, WDR5 0103, WDR5-0103, inhibit, Histone Methyltransferase, WDR-5-0103, WD-Repeat Protein 5-0103

WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd: 450 nM).

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

WDR5-0103, CAS 890190-22-4

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd: 450 nM).
Targets&IC50	WDR5:450 nM

Synonyms	WDR50103, Inhibitor, WDR5 0103, WDR5-0103, inhibit, Histone Methyltransferase, WDR-5-0103, WD-Repeat Protein 5-0103
Molecular Weight	383.448
Formula	C21H25N3O4
CAS No.	890190-22-4

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 40 mg/mL

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Senisterra G, et al. Biochem J. 2013 Jan 1;449(1):151-9.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Compound Library Anti-Pancreatic Cancer Compound Library Inhibitor Library Histone Modification Compound Library Immunology/Inflammation Compound Library Kinase Inhibitor Library Stem Cell Differentiation Compound Library Epigenetics Compound Library Angiogenesis related Compound Library JAK-STAT Compound Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.