Shopping Cart
- Remove All
![TargetMol](https://newstatic.targetmol.com/error/oops.webp)
Your shopping cart is currently empty
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $327 | In Stock | |
2 mg | $492 | In Stock | |
5 mg | $737 | In Stock | |
10 mg | $1,110 | In Stock | |
25 mg | $1,650 | In Stock | |
50 mg | $2,230 | In Stock | |
100 mg | $2,930 | In Stock |
Description | [(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31. [(pF)Phe4]Nociceptin(1-13)NH2 acetate displays high selectivity over δ, κ, and μ opioid receptors (>3000 fold). |
In vivo | In unanaesthetised normotensive mice, [(pF)Phe4]Nociceptin(1-13)NH2 acetate (100 nmol/kg; i.c.v.) dose-dependently stimulated feeding in rats and is about tenfold more potent than NC(1-13)NH2. [(pF)Phe4]Nociceptin(1-13)NH2 acetate (100 nmol/kg; i.v.) decreases mean blood pressure and heart rate; these effects are longer lasting than those elicited by the same dose of NC(1-13)NH2[1]. |
Molecular Weight | 1459.63 |
Formula | C63H103FN22O17 |
Cas No. |
Storage | keep away from moisture Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.