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BMS-195270
Catalog No. T30503Cas No. 202822-23-9
BMS-195270 is a tissue-specific inhibitor of bladder muscle tone and spontaneous contraction in rats. It can inhibit Carbachol-induced tone and inhibit calcium flux in isolated rat bladder tissue strips in an isolated bladder model.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $59 | In Stock | |
| 5 mg | $143 | In Stock | |
| 10 mg | $228 | In Stock | |
| 25 mg | $463 | In Stock | |
| 50 mg | $745 | In Stock | |
| 100 mg | $987 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | BMS-195270 is a tissue-specific inhibitor of bladder muscle tone and spontaneous contraction in rats. It can inhibit Carbachol-induced tone and inhibit calcium flux in isolated rat bladder tissue strips in an isolated bladder model. |
| In vitro | BMS-195270 inhibited the response of HEK293 cells to the muscarinic agonist carbachol (the EC50 was 2 μM)[1]. |
| Alias | UNII-20UM0T170J, BMS 195270, BMS195270, CHEMBL13637, SCHEMBL5754043 |
| Molecular Weight | 355.7 |
| Formula | C15H9ClF3N3O2 |
| Cas No. | 202822-23-9 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 100 mg/mL (281.14 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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