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CDD0102
😃Good
Catalog No. T10731Cas No. 146422-58-4
Alias CDD0102A
CDD0102 is a potent agonist of M1 Muscarinic receptor.
CDD0102
😃Good
Catalog No. T10731Alias CDD0102ACas No. 146422-58-4
CDD0102 is a potent agonist of M1 Muscarinic receptor.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,520 | 6-8 weeks | |
| 50 mg | $1,980 | 6-8 weeks | |
| 100 mg | $2,500 | 6-8 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | CDD0102 is a potent agonist of M1 Muscarinic receptor. |
| In vitro | CDD0102 displays much lower activity at M3 and M5 receptors. |
| In vivo | CDD0102 (i.p.) crosses the blood-brain barrier (BBB) in a dose-dependent manner. In toxicological studies, the LD50 of CDD0102 is 190 mg/kg following i.p. injections and greater than 1,000 mg/kg following oral administration. CDD0102 (10 mg/kg) fully reverses memory deficits associated with IgG-192 saporin administration. Again, no side effects are observed at this dose. |
| Alias | CDD0102A |
| Molecular Weight | 180.21 |
| Formula | C8H12N4O |
| Cas No. | 146422-58-4 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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