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CGP 36742
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Catalog No. T14938Cas No. 123690-78-8
Alias SGS-742
CGP 36742 is a selective antagonist of the GABAB receptor that can penetrate the blood-brain barrier after peripheral administration (IC50: 32 μM). It is useful in the treatment of depression.
CGP 36742
😃Good
Catalog No. T14938Alias SGS-742Cas No. 123690-78-8
CGP 36742 is a selective antagonist of the GABAB receptor that can penetrate the blood-brain barrier after peripheral administration (IC50: 32 μM). It is useful in the treatment of depression.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $83 | 5 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | CGP 36742 is a selective antagonist of the GABAB receptor that can penetrate the blood-brain barrier after peripheral administration (IC50: 32 μM). It is useful in the treatment of depression. |
| Targets&IC50 | GABAB:32 μM |
| Alias | SGS-742 |
| Molecular Weight | 179.2 |
| Formula | C7H18NO2P |
| Cas No. | 123690-78-8 |
| Relative Density. | 1.057 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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