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Enerisant
🥰Excellent
Catalog No. T67828Cas No. 1152747-82-4
Alias TS-091
Enerisant (TS-091) is an orally active, selective and potent histamine H3 receptor antagonist that modulates histamine H3 receptors in mice in a dose-dependent manner.Enerisant promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.
Enerisant
🥰Excellent
Purity: 99.7%
Catalog No. T67828Alias TS-091Cas No. 1152747-82-4
Enerisant (TS-091) is an orally active, selective and potent histamine H3 receptor antagonist that modulates histamine H3 receptors in mice in a dose-dependent manner.Enerisant promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 93 € | In Stock | |
| 5 mg | 215 € | In Stock | |
| 10 mg | 346 € | In Stock | |
| 25 mg | 730 € | In Stock | |
| 50 mg | 1.168 € | In Stock | |
| 100 mg | 1.871 € | In Stock | |
| 1 mL x 10 mM (in DMSO) | 188 € | In Stock |
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Purity:99.7%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Enerisant (TS-091) is an orally active, selective and potent histamine H3 receptor antagonist that modulates histamine H3 receptors in mice in a dose-dependent manner.Enerisant promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits. |
| Targets&IC50 | H3 receptor (rat):14.5 nM, H3 receptor (rat):7.87 nM, H3 receptor (human):2.89 nM, H3 receptor (human):1.65 nM（Ki） |
| In vivo | In the male SD rat model of R-α-methylhistamine-induced dipsogenia, Enerisant (oral, single dose, 0.1, 0.3, and 1 mg/kg) attenuated the dipsogenic response[1]. |
| Alias | TS-091 |
| Molecular Weight | 398.50 |
| Formula | C22H30N4O3 |
| Cas No. | 1152747-82-4 |
| Smiles | C(=O)(C1=CN(N=C1)C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N4CCOCC4 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (200.75 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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