Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

GSK251

🥰Excellent
Catalog No. T39573Cas No. 2125968-05-8

GSK251 is a novel, orally bioavailable inhibitor of PI3Kδ, exhibiting high potency and selectivity, with a unique binding mode.

GSK251

GSK251

🥰Excellent
Purity: 98.9%
Catalog No. T39573Cas No. 2125968-05-8
GSK251 is a novel, orally bioavailable inhibitor of PI3Kδ, exhibiting high potency and selectivity, with a unique binding mode.
Pack SizePriceAvailabilityQuantity
1 mg157 €In Stock
5 mg396 €In Stock
10 mg562 €In Stock
25 mg837 €In Stock
50 mg1.121 €In Stock
100 mg1.520 €In Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "GSK251"

Select Batch
Purity:98.9%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
GSK251 is a novel, orally bioavailable inhibitor of PI3Kδ, exhibiting high potency and selectivity, with a unique binding mode.
Chemical Properties
Molecular Weight584.71
FormulaC29H37FN6O4S
Cas No.2125968-05-8
SmilesCOc1ncc(cc1S(=O)(=O)Nc1ccnc(c1)-c1ccc(CN2CCN(CC2)C(C)C)cc1F)N1CCOCC1
Relative Density.1.295 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 50 mg/mL (85.5 mM), Sonication and heating to 60℃ are recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.7102 mL8.5512 mL17.1025 mL85.5125 mL
5 mM0.3420 mL1.7102 mL3.4205 mL17.1025 mL
10 mM0.1710 mL0.8551 mL1.7102 mL8.5512 mL
20 mM0.0855 mL0.4276 mL0.8551 mL4.2756 mL
50 mM0.0342 mL0.1710 mL0.3420 mL1.7102 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy GSK251 | purchase GSK251 | GSK251 cost | order GSK251 | GSK251 chemical structure | GSK251 formula | GSK251 molecular weight