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Odapipam
Catalog No. T12288Cas No. 131796-63-9
Alias NNC 756
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
Odapipam
Catalog No. T12288Alias NNC 756Cas No. 131796-63-9
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,220 | 6-8 weeks | |
| 50 mg | $1,590 | 6-8 weeks | |
| 100 mg | $2,430 | 6-8 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM). |
| In vivo | The metabolic pathway of Odapipam in phenobarbital-induced rat liver microsomes has been examined, revealing the formation of five distinct metabolites during its incubation. Analysis of the electron-ionization (EI+) mass spectra identified these metabolites as N-desmethyl-Odapipam, 1-hydroxy-Odapipam, two isomers of 3′-hydroxy-Odapipam, and a dehydrogenated metabolite within the dihydrobenzofuran moiety[1]. |
| Alias | NNC 756 |
| Molecular Weight | 329.82 |
| Formula | C19H20ClNO2 |
| Cas No. | 131796-63-9 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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