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Regadenoson

🥰Excellent
Catalog No. T2671Cas No. 313348-27-5
Alias Lexiscan, CVT-3146

Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine receptor, which induces coronary vasodilation. This leads to an increase in coronary blood flow and enhances myocardial perfusion. Compared to adenosine, regadenoson has a longer half-life and shows higher selectivity towards the A2A adenosine receptor. This agent is a very weak agonist for the A1 adenosine receptor and has negligible affinity for the A2B and A3 adenosine receptors.

Regadenoson

Regadenoson

🥰Excellent
Purity: 100%
Catalog No. T2671Alias Lexiscan, CVT-3146Cas No. 313348-27-5
Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine receptor, which induces coronary vasodilation. This leads to an increase in coronary blood flow and enhances myocardial perfusion. Compared to adenosine, regadenoson has a longer half-life and shows higher selectivity towards the A2A adenosine receptor. This agent is a very weak agonist for the A1 adenosine receptor and has negligible affinity for the A2B and A3 adenosine receptors.
Pack SizePriceAvailabilityQuantity
2 mg$39In Stock
5 mg$59In Stock
10 mg$93In Stock
25 mg$183In Stock
50 mg$287In Stock
100 mg$438In Stock
500 mg$985In Stock
1 mL x 10 mM (in DMSO)$66In Stock
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Purity:100%
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Product Introduction

Bioactivity
Description
Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine receptor, which induces coronary vasodilation. This leads to an increase in coronary blood flow and enhances myocardial perfusion. Compared to adenosine, regadenoson has a longer half-life and shows higher selectivity towards the A2A adenosine receptor. This agent is a very weak agonist for the A1 adenosine receptor and has negligible affinity for the A2B and A3 adenosine receptors.
Targets&IC50
A2AR:290 nM(Ki)
AliasLexiscan, CVT-3146
Chemical Properties
Molecular Weight390.35
FormulaC15H18N8O5
Cas No.313348-27-5
SmilesCNC(=O)c1cnn(c1)-c1nc(N)c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Relative Density.1.98g/cm3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 9 mg/mL (23.06 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.5618 mL12.8090 mL25.6180 mL128.0902 mL
5 mM0.5124 mL2.5618 mL5.1236 mL25.6180 mL
10 mM0.2562 mL1.2809 mL2.5618 mL12.8090 mL
20 mM0.1281 mL0.6405 mL1.2809 mL6.4045 mL

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