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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $34 | In Stock | |
5 mg | $80 | In Stock | |
10 mg | $128 | In Stock | |
25 mg | $289 | In Stock | |
50 mg | $455 | In Stock | |
100 mg | $672 | In Stock | |
500 mg | $1,430 | In Stock |
Description | TASK-1-IN-1 is a potent and selective inhibitor of TASK-1 (Potassium Channel) with an IC50 of 148 nM, and exhibits a reduced inhibitory effect on the TASK-3 channel with an IC50 of 1750 nM. TASK-1-IN-1 also demonstrates anticancer effects. |
Targets&IC50 | TASK1:148 nM, TASK3:1750 nM |
In vitro | TASK-1-IN-1 (compound F3) inhibits cell proliferation and viability in MCF-7 cancer cells. This effect is absent in TASK-1 knockdown MCF-7 cells, indicating its specificity for TASK-1 channels.[1] |
Molecular Weight | 344.41 |
Formula | C22H20N2O2 |
Cas No. | 600125-11-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO: < 1 mg/mL (insoluble) ![]() |
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