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1-Ethynylpyrene
Catalog No. T9704Cas No. 34993-56-1
1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $39 | In Stock | |
| 10 mg | $64 | In Stock | |
| 25 mg | $107 | In Stock | |
| 50 mg | $163 | In Stock | |
| 100 mg | $278 | In Stock | |
| 200 mg | $418 | In Stock | |
| 500 mg | $682 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $44 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | 1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM). |
| In vitro | The Ki values of 1-Ethynylpyrene against P450 1A2, and 2B1 is 0.32 and 0.04 μM, respectively[1]. |
| Molecular Weight | 226.27 |
| Formula | C18H10 |
| Cas No. | 34993-56-1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||
| Solubility Information | DMSO: 3.06 mg/mL (13.5 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
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