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1-Stearoyl-2-arachidonoyl-sn-glycerol
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Catalog No. T40757Cas No. 65914-84-3
1-Stearoyl-2-arachidonoyl-sn-glycerol (DAG) is a diacylglycerol (DAG) substrate that can be hydrolyzed to 2-arachidonic acid glycerol. 1-Stearoyl-2-arachidonoyl-sn-glycerol activates PKC, induces Ca2+ influx, and can induce tracheal smooth muscle contraction.
1-Stearoyl-2-arachidonoyl-sn-glycerol
😃Good
Catalog No. T40757Cas No. 65914-84-3
1-Stearoyl-2-arachidonoyl-sn-glycerol (DAG) is a diacylglycerol (DAG) substrate that can be hydrolyzed to 2-arachidonic acid glycerol. 1-Stearoyl-2-arachidonoyl-sn-glycerol activates PKC, induces Ca2+ influx, and can induce tracheal smooth muscle contraction.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg (15.50 mM * 5 μL in Methyl acetate) | $645 | 35 days | |
| 10 mg (15.50 mM * 1 mL in Methyl acetate) | $1,210 | 35 days | |
| 25 mg (15.50 mM * 2.5 mL in Methyl acetate) | $2,630 | 35 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | 1-Stearoyl-2-arachidonoyl-sn-glycerol (DAG) is a diacylglycerol (DAG) substrate that can be hydrolyzed to 2-arachidonic acid glycerol. 1-Stearoyl-2-arachidonoyl-sn-glycerol activates PKC, induces Ca2+ influx, and can induce tracheal smooth muscle contraction. |
| In vitro | 1-Stearoyl-2-arachidonoyl-sn-glycerol (0.3-3 μM) enhances non-selective cation channel (NSCC) activity in airway smooth muscle cells; 1-Stearoyl-2-arachidonoyl-sn-glycerol (0-5 μM) It has a significant stimulating effect on the activation of PKCα, PKCδ, PKCγ, PKCε and PKCβI [2]. |
| Molecular Weight | 645.01 |
| Formula | C41H72O5 |
| Cas No. | 65914-84-3 |
| Smiles | [C@@H](OC(CCC/C=C\C/C=C\C/C=C\C/C=C\CCCCC)=O)(COC(CCCCCCCCCCCCCCCCC)=O)CO |
| Relative Density. | 0.942g/cm3 |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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