Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 55.00 | |
10 mg | In stock | $ 80.00 | |
25 mg | In stock | $ 129.00 | |
50 mg | In stock | $ 187.00 | |
100 mg | In stock | $ 247.00 | |
200 mg | In stock | $ 372.00 | |
500 mg | In stock | $ 629.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 67.00 |
Description | Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). |
Targets&IC50 | Ghrelin receptor:(EC50)0.74 nM , Ghrelin receptor:(ki)0.7 nM |
In vitro | Anamorelin(ANAM) is a potent and highly specific ghrelin receptor agonist |
In vivo | Anamorelin(ANAM) showed significant agonist and binding activity on the ghrelin receptor, and stimulated GH release in vitro.?In rats, ANAM significantly and dose-dependently increased FI and BW at all dose levels compared with control, and significantly increased GH levels at 10 or 30 mg/kg doses.?Increases in GH and IGF-1 levels were observed following ANAM administration in pigs. |
Synonyms | RC-1291, ONO-7643 |
Molecular Weight | 546.7 |
Formula | C31H42N6O3 |
CAS No. | 249921-19-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (182.92 mM)
You can also refer to dose conversion for different animals. More
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Anamorelin 249921-19-5 GPCR/G Protein GHSR Growth hormone secretagogue receptor RC-1291 Inhibitor RC 1291 ONO7643 ONO 7643 ONO-7643 RC1291 inhibit inhibitor