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AnaMorelin hydrochloride

Catalog No. T7225Cas No. 861998-00-7
Alias RC-1291 hydrochloride, ONO-7643 hydrochloride

AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).

AnaMorelin hydrochloride

AnaMorelin hydrochloride

Purity: 99.18%
Catalog No. T7225Alias RC-1291 hydrochloride, ONO-7643 hydrochlorideCas No. 861998-00-7
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
Pack SizePriceAvailabilityQuantity
1 mg$30In Stock
2 mg$43In Stock
5 mg$67In Stock
10 mg$97In Stock
25 mg$148In Stock
50 mg$187In Stock
100 mg$247In Stock
1 mL x 10 mM (in DMSO)$87In Stock
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Purity:99.18%
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Product Introduction

Bioactivity
Description
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
Targets&IC50
Ghrelin receptor (FLIPR assay):0.74 nM(EC50)
In vivo
In rats, AnaMorelin hydrochloride(ANAM) significantly and dose-dependently increased FI and BW at all dose levels compared with control, and significantly increased GH levels at 10 or 30 mg/kg doses. Increases in GH and IGF-1 levels were observed following ANAM administration in pigs[1].
Animal Research
Fluorescent imaging plate reader and binding assays in HEK293 and baby hamster kidney cells determined the agonist and antagonist activity of ANAM, and its affinity for the ghrelin receptor. Rat pituitary cells were incubated with ANAM to evaluate its effect on growth hormone (GH) release. In vivo, rats were treated with ANAM 3, 10, or 30 mg/kg, or control orally, once daily for 6 days to evaluate the effect on food intake (FI) and body weight (BW), and once to assess GH response. In pigs, single (3.5 mg/kg) or continuous (1 mg/kg/day) ANAM doses were administered to assess GH and insulin-like growth factor (IGF-1) response[1].
AliasRC-1291 hydrochloride, ONO-7643 hydrochloride
Chemical Properties
Molecular Weight583.16
FormulaC31H43ClN6O3
Cas No.861998-00-7
Storage & Solubility Information
Storagestore at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 28 mg/mL (48.01 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.7148 mL8.5740 mL17.1480 mL85.7398 mL
5 mM0.3430 mL1.7148 mL3.4296 mL17.1480 mL
10 mM0.1715 mL0.8574 mL1.7148 mL8.5740 mL
20 mM0.0857 mL0.4287 mL0.8574 mL4.2870 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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