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AnaMorelin hydrochloride
🥰Excellent
Catalog No. T7225Cas No. 861998-00-7
Alias RC-1291 hydrochloride, ONO-7643 hydrochloride
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
AnaMorelin hydrochloride
🥰Excellent
Purity: 99.18%
Catalog No. T7225Alias RC-1291 hydrochloride, ONO-7643 hydrochlorideCas No. 861998-00-7
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $30 | In Stock | |
| 2 mg | $43 | In Stock | |
| 5 mg | $67 | In Stock | |
| 10 mg | $97 | In Stock | |
| 25 mg | $148 | In Stock | |
| 50 mg | $187 | In Stock | |
| 100 mg | $247 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $87 | In Stock |
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Purity:99.18%
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With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.Product Introduction
Bioactivity
Chemical Properties
| Description | AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay). |
| Targets&IC50 | Ghrelin receptor (FLIPR assay):0.74 nM(EC50) |
| In vivo | In rats, AnaMorelin hydrochloride(ANAM) significantly and dose-dependently increased FI and BW at all dose levels compared with control, and significantly increased GH levels at 10 or 30 mg/kg doses. Increases in GH and IGF-1 levels were observed following ANAM administration in pigs[1]. |
| Animal Research | Fluorescent imaging plate reader and binding assays in HEK293 and baby hamster kidney cells determined the agonist and antagonist activity of ANAM, and its affinity for the ghrelin receptor. Rat pituitary cells were incubated with ANAM to evaluate its effect on growth hormone (GH) release. In vivo, rats were treated with ANAM 3, 10, or 30 mg/kg, or control orally, once daily for 6 days to evaluate the effect on food intake (FI) and body weight (BW), and once to assess GH response. In pigs, single (3.5 mg/kg) or continuous (1 mg/kg/day) ANAM doses were administered to assess GH and insulin-like growth factor (IGF-1) response[1]. |
| Alias | RC-1291 hydrochloride, ONO-7643 hydrochloride |
| Molecular Weight | 583.16 |
| Formula | C31H43ClN6O3 |
| Cas No. | 861998-00-7 |
| Smiles | Cl.[H][C@](Cc1c[nH]c2ccccc12)(NC(=O)C(C)(C)N)C(=O)N1CCC[C@@](Cc2ccccc2)(C1)C(=O)N(C)N(C)C |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 28 mg/mL (48.01 mM) | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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