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CID 2745687

Catalog No. T21874   CAS 264233-05-8

CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two agonists that share an overlapping binding site.

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CID 2745687 Chemical Structure
CID 2745687, CAS 264233-05-8
Pack Size Availability Price/USD Quantity
1 mg In stock $ 34.00
2 mg In stock $ 48.00
5 mg In stock $ 80.00
10 mg In stock $ 128.00
25 mg In stock $ 289.00
50 mg In stock $ 455.00
100 mg In stock $ 672.00
1 mL * 10 mM (in DMSO) In stock $ 89.00
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Purity: 99.11%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two agonists that share an overlapping binding site.
Molecular Weight 395.43
Formula C17H19F2N5O2S
CAS No. 264233-05-8

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 60 mg/ml (151.73 mM)

TargetMolReferences and Literature

1. Jenkins L , Harries N , Lappin J E , et al. Antagonists of GPR35 display high species ortholog selectivity and varying modes of action[J]. Journal of Pharmacology & Experimental Therapeutics, 2012, 343(3):683-695.

Related compound libraries

This product is contained In the following compound libraries:
GPCR Compound Library Endocrinology-Hormone Compound Library NO PAINS Compound Library Inhibitor Library Bioactive Compounds Library Max Bioactive Compound Library

Related Products

Related compounds with same targets
Tyrphostin A25 Kisspeptin 234 acetate(1145998-81-7 free base) APD668 SNAP 94847 YUM70 RTI-13951-33 GPR35 agonist 2 PW0787

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Keywords

CID 2745687 264233-05-8 Endocrinology/Hormones GPCR/G Protein GPR GPCR G Protein-coupled Receptors inhibit CID2745687 Inhibitor Arrestin GPR35 antagonist CID-2745687 inhibitor

 

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