Powder: -20°C for 3 years | In solvent: -80°C for 1 year
dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and inactive on BRD4BD2
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 48.00 | |
2 mg | In stock | $ 67.00 | |
5 mg | In stock | $ 122.00 | |
10 mg | In stock | $ 189.00 | |
25 mg | In stock | $ 293.00 | |
50 mg | In stock | $ 455.00 | |
100 mg | In stock | $ 672.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 178.00 |
Description | dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and inactive on BRD4BD2 |
Targets&IC50 | BRD4 BD1:500 nM (DC50) |
Molecular Weight | 699.18 |
Formula | C34H31ClN8O5S |
CAS No. | 1883863-52-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (357.56 mM)
You can also refer to dose conversion for different animals. More
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Dbet57 1883863-52-2 Chromatin/Epigenetic Epigenetic Reader Domain inhibit Dbet-57 dBET 57 Inhibitor PROTACs inhibitor