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JNJ-38158471

JNJ-38158471
JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor with IC50 of 40 nM, inhibits closely related tyrosine kinases such as Ret and Kit with IC50 of 180 nM and 500 nM.
Catalog No. T22349Cas No. 951151-97-6
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Purity:97.08%
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JNJ-38158471

Catalog No. T22349Cas No. 951151-97-6
JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor with IC50 of 40 nM, inhibits closely related tyrosine kinases such as Ret and Kit with IC50 of 180 nM and 500 nM.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Pack SizePriceAvailabilityQuantity
1 mg$48In Stock
2 mg$68In Stock
5 mg$107In Stock
10 mg$158In Stock
25 mg$273In Stock
50 mg$397In Stock
100 mg$535In Stock
200 mg$735In Stock
1 mL x 10 mM (in DMSO)$115In Stock
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Product Introduction

Bioactivity
Description
JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor with IC50 of 40 nM, inhibits closely related tyrosine kinases such as Ret and Kit with IC50 of 180 nM and 500 nM.
Targets&IC50
VEGFR2:40 nM
AliasCS-2660
Chemical Properties
Molecular Weight364.79
FormulaC15H17ClN6O3
Cas No.951151-97-6
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 30 mg/ml (82.24 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.7413 mL13.7065 mL27.4130 mL137.0652 mL
5 mM0.5483 mL2.7413 mL5.4826 mL27.4130 mL
10 mM0.2741 mL1.3707 mL2.7413 mL13.7065 mL
20 mM0.1371 mL0.6853 mL1.3707 mL6.8533 mL
50 mM0.0548 mL0.2741 mL0.5483 mL2.7413 mL

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