Powder: -20°C for 3 years | In solvent: -80°C for 1 year
LY2922470 is a potent, selective G protein-coupled receptor 40 (GPR40) agonist, with EC50s of 7 nM for human GPR40, 1 nM for mouse GPR40 and 3 nM for rat GPR40, respectively. LY2922470 reduces glucose levels along and increases insulin and GLP-1 significantly.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 117.00 | |
5 mg | In stock | $ 249.00 | |
10 mg | In stock | $ 374.00 | |
25 mg | In stock | $ 649.00 | |
50 mg | In stock | $ 926.00 | |
100 mg | In stock | $ 1,260.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 261.00 |
Description | LY2922470 is a potent, selective G protein-coupled receptor 40 (GPR40) agonist, with EC50s of 7 nM for human GPR40, 1 nM for mouse GPR40 and 3 nM for rat GPR40, respectively. LY2922470 reduces glucose levels along and increases insulin and GLP-1 significantly. |
Targets&IC50 | FFA1/GPR40:1 nM(EC50,mouse), FFA1/GPR40:3 nM(EC50,rat), FFA1/GPR40:7 nM(EC50, human) |
Molecular Weight | 475.6 |
Formula | C28H29NO4S |
CAS No. | 1423018-12-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 125 mg/mL (262.83 mM)
You can also refer to dose conversion for different animals. More
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LY2922470 1423018-12-5 Endocrinology/Hormones GPCR/G Protein GPR Free Fatty Acid Receptor inhibit Inhibitor FFAR LY-2922470 LY 2922470 inhibitor