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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $79 | In Stock | |
5 mg | $165 | In Stock | |
10 mg | $235 | In Stock | |
25 mg | $419 | In Stock | |
50 mg | $598 | In Stock | |
100 mg | $853 | In Stock | |
1 mL x 10 mM (in DMSO) | $168 | In Stock |
Description | S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors. |
Kinase Assay | PI3K inhibition by LY294002 is determined in a radiometric assay using purified, recombinant enzymes with 1 μM ATP. The kinase reaction is carried out for 1 hour at room temperature (24oC) and is terminated by addition of PBS. IC50 values are subsequently determined using a sigmoidal dose-response curve fit (variable slope). CK2 and GSK3β (glycogen synthase kinase 3β) inhibition are established by kinase selectivity screening. LY294002 is tested against the Upstate panel of kinases in 10 μM ATP.[4] |
Molecular Weight | 324.85 |
Formula | C17H25ClN2O2 |
Cas No. | 1222097-72-4 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
Solubility Information | DMSO: 25 mg/mL (76.96 mM) ![]() | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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