Shopping Cart
- Remove All
- Your shopping cart is currently empty
VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK, Kir3) activator.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | 53 € | In Stock | |
5 mg | 130 € | In Stock | |
10 mg | 207 € | In Stock | |
25 mg | 348 € | In Stock | |
50 mg | 466 € | In Stock | |
100 mg | 620 € | In Stock | |
200 mg | 843 € | In Stock | |
1 mL x 10 mM (in DMSO) | 144 € | In Stock |
Description | VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK, Kir3) activator. |
Targets&IC50 | GIRK1/2:165 nM(EC50) , GIRK1/4:720 nM(EC50) |
In vivo | Reduced stress‐induced hyperthermia (SIH), a physiological test of anxiolytic efficacy in wild mice, but had no impact in and Kcnj3 (Girk1) ?/? mice. |
Animal Research | Animal Model:Male C57BL/6J mice, Kcnj3?/? siblings female and male C57BL/6J mice. Dosage:10 mg/kg; 30mg/kg. Administration:Intraperitoneal injection |
Molecular Weight | 349.83 |
Formula | C18H21ClFN3O |
Cas No. | 2126040-21-7 |
Smiles | Cc1cc(NC(=O)Cc2ccc(F)c(Cl)c2)n(n1)C1CCCCC1 |
Relative Density. | 1.31 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 250 mg/mL (714.63 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
|
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.