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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $453 | In Stock | |
5 mg | $913 | In Stock | |
10 mg | $1,319 | In Stock | |
25 mg | $2,090 | In Stock | |
1 mL x 10 mM (in DMSO) | $1,190 | In Stock |
Description | C-82 is a specific CBP/β-catenin antagonist. It inhibits the binding between β-catenin and CBP and increases the binding between β-catenin and p300. |
In vitro | C-82 inhibits the activation of isolated primary mouse quiescent hepatic stellate cells (HSCs) and promotes cell death in culture-activated HSCs. |
In vivo | PRI-724 is phosphorylated-C-82 and is rapidly hydrolyzed to its active form C-82 in vivo, and pre-clinical studies have shown a very acceptable toxicity profile. |
Molecular Weight | 578.66 |
Formula | C33H34N6O4 |
Cas No. | 1422253-37-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
Solubility Information | DMSO: 55 mg/ml (95.05 mM) ![]() | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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