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CaMKP Inhibitor

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Purity:99.98%

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COA LCMS HNMR

CaMKP Inhibitor

Catalog No. T2159Cas No. 52789-62-5

CaMKP Inhibitor can inhibit CaMKP.

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Pack Size	Price	Availability
1 mg	$35	In Stock
5 mg	$79	In Stock
10 mg	$129	In Stock
25 mg	$253	In Stock
50 mg	$371	In Stock
100 mg	$512	In Stock
500 mg	$1,150	In Stock
1 mL x 10 mM (in DMSO)	$109	In Stock

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Product Introduction

Bioactivity

Description

CaMKP Inhibitor can inhibit CaMKP.

Kinase Assay

Biacore study: Competition assay is performed on a Biacore S51. A Series S Sensor chip CM5 is utilized for the immobilization of a PentaHis antibody for capture of the His-tagged p53. The level of capture is ~200 response units (1 response unit corresponds to 1 pg of protein per mm 2). The concentration of MDM2 protein is kept constant at 300 nM. Nutlin-3 is dissolved in DMSO at 10 mM and further diluted to make a concentration series of Nutlin-3 in each MDM2 test sample. The assay is run at 25°C in running buffer (10 mM Hepes, 0.15 M NaCl, 2% DMSO). MDM2-p53 binding in the presence of Nutlin-3 is calculated as a percentage of binding in the absence of Nutlin-3 and IC50 is calculated

Chemical Properties

Molecular Weight	341.28
Formula	C10H8NNaO7S2
Cas No.	52789-62-5

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 34.48 mg/mL (101.04 mM)

DMSO: 10 mM

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9301 mL	14.6507 mL	29.3015 mL	146.5073 mL
5 mM	0.5860 mL	2.9301 mL	5.8603 mL	29.3015 mL

H2O

	1mg	5mg	10mg	50mg
10 mM	0.2930 mL	1.4651 mL	2.9301 mL	14.6507 mL
20 mM	0.1465 mL	0.7325 mL	1.4651 mL	7.3254 mL
50 mM	0.0586 mL	0.2930 mL	0.5860 mL	2.9301 mL
100 mM	0.0293 mL	0.1465 mL	0.2930 mL	1.4651 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

You can also refer to dose conversion for different animals. More

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc