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CDK9-IN-1
🥰Excellent
Catalog No. T10741Cas No. 1415559-43-1
CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.
CDK9-IN-1
🥰Excellent
Purity: 98.52%
Catalog No. T10741Cas No. 1415559-43-1
CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $128 | In Stock | |
| 5 mg | $189 | In Stock |
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Purity:98.52%
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Product Introduction
Bioactivity
Chemical Properties
| Description | CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections. |
| Targets&IC50 | CDK9-CyclinT1:39 nM |
| In vitro | CDK9-IN-1 is a selective CDK9 inhibitor with an IC50 = 39 nM for CDK9/CycT1. p24 analysis of CDK9-IN-1 revealed that it can be used for the treatment of HIV infection. [1] |
| Molecular Weight | 499.54 |
| Formula | C26H21N5O4S |
| Cas No. | 1415559-43-1 |
| Smiles | O=C1C=2C=CC=CC2C(=O)N1C3=CC=CC(=C3)C=4N=CN=C(C4)NC5=CC=C(C(=C5)NS(=O)(=O)C)C |
| Relative Density. | 1.463 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL(160.15 mM), Sonication is recommended. H2O: < 0.1 mg/mL (insoluble) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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