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DPCPX
Catalog No. T22744Cas No. 102146-07-6
Alias PD 116948
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
DPCPX
Catalog No. T22744Alias PD 116948Cas No. 102146-07-6
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $41 | In Stock | |
| 25 mg | $65 | In Stock | |
| 50 mg | $98 | In Stock | |
| 100 mg | $144 | In Stock |
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Purity:99.93%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | DPCPX (PD 116948) is an A1 adenosine receptor antagonist |
| Targets&IC50 | [3H]-CHA binding to A1 receptor (rat whole brain membranes):0.46 nM (Ki), [3H]-NECA binding to A2 receptor (rat striatal membranes):340 nM (Ki) |
| In vivo | DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine, escitalopram, and reboxetine in mice behavioral tests |
| Alias | PD 116948 |
| Molecular Weight | 304.39 |
| Formula | C16H24N4O2 |
| Cas No. | 102146-07-6 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | Ethanol: < 1 mg/mL (insoluble or slightly soluble) DMSO: 3.04 mg/ml (10 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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