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Flovagatran
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Catalog No. T31806Cas No. 871576-03-3
Alias TGN 255
Flovagatran (TGN 255) is an orally active, potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.
Flovagatran
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Purity: 99.56%
Catalog No. T31806Alias TGN 255Cas No. 871576-03-3
Flovagatran (TGN 255) is an orally active, potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $762 | In Stock | |
| 5 mg | $1,590 | In Stock | |
| 10 mg | $1,980 | In Stock | |
| 50 mg | $2,580 | 6-8weeks |
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Purity:99.56%
ee:98.92%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Flovagatran (TGN 255) is an orally active, potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism. |
| In vivo | Flovagatran (2.5-mg/kg bolus plus 10 mg/kg/h for 90 minutes) induces anticoagulation effects in dogs [1]. |
| Alias | TGN 255 |
| Molecular Weight | 525.4 |
| Formula | C27H36BN3O7 |
| Cas No. | 871576-03-3 |
| Smiles | C([C@@H](CC1=CC=CC=C1)NC(OCC2=CC=CC=C2)=O)(=O)N3[C@H](C(N[C@@H](CCCOC)B(O)O)=O)CCC3 |
| Relative Density. | 1.237 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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