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Gentisin
🥰Excellent
Catalog No. TN1683Cas No. 437-50-3
Gentisin is a novel inhibitor of vascular smooth muscle cells (VSMC) proliferation with an IC50 value of 7.84 μM. Gentisin has mutagenic activity.
Gentisin
🥰Excellent
Purity: 95.34%
Catalog No. TN1683Cas No. 437-50-3
Gentisin is a novel inhibitor of vascular smooth muscle cells (VSMC) proliferation with an IC50 value of 7.84 μM. Gentisin has mutagenic activity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 100 € | In Stock | |
| 5 mg | 248 € | In Stock | |
| 10 mg | 369 € | In Stock | |
| 25 mg | 606 € | In Stock | |
| 50 mg | 837 € | In Stock | |
| 1 mL x 10 mM (in DMSO) | 227 € | In Stock |
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Purity:95.34%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Gentisin is a novel inhibitor of vascular smooth muscle cells (VSMC) proliferation with an IC50 value of 7.84 μM. Gentisin has mutagenic activity. |
| Targets&IC50 | VSMC cells:7.84 μM |
| In vitro | The anti-proliferative effect of Gentisin was confirmed by the quantification of DNA synthesis (BrdU incorporation) in VSMC. Cell death quantification (determined by LDH release in the culture medium) revealed that Gentisin was not cytotoxic in the investigated concentration range[1]. |
| Molecular Weight | 258.23 |
| Formula | C14H10O5 |
| Cas No. | 437-50-3 |
| Smiles | COc1cc(O)c2c(c1)oc1ccc(O)cc1c2=O |
| Relative Density. | 1.3326 g/cm3 (Estimated) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (309.80 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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