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GR 94800 acetate

🥰Excellent
Catalog No. T22811L
Alias GR 94800 acetate (141636-65-9 free base)

GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.

GR 94800 acetate

GR 94800 acetate

🥰Excellent
Purity: 97.86%
Catalog No. T22811LAlias GR 94800 acetate (141636-65-9 free base)
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Pack SizePriceAvailabilityQuantity
1 mg$382In Stock
2 mg$542In Stock
5 mg$816In Stock
10 mg$1,090In Stock
25 mg$1,630In Stock
50 mg$2,200In Stock
100 mg$2,970In Stock
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Purity:97.86%
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Product Introduction

Bioactivity
Description
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Targets&IC50
NK3:6.0(pKb), NK1:6.4(pKb), NK2:9.6(pKb)
In vitro
GR 94800 displayed high affinity (pIC50 8.4-9.5) with no significant difference in potency between these four tissues from the rat fundus, colon, bladder and vas deferens[3].
AliasGR 94800 acetate (141636-65-9 free base)
Chemical Properties
Molecular Weight964.12
FormulaC51H65N9O10
SmilesCCCC[C@@H](C(N)=O)NC([C@H](CCC1)N1C([C@@H](CCC1)N1C([C@H](Cc1ccccc1)NC([C@@H](Cc1c[nH]c2c1cccc2)NC([C@H](C)NC([C@H](C)NC(c1ccccc1)=O)=O)=O)=O)=O)=O)=O.CC(O)=O
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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