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JNJ-39220675
🥰Excellent
Catalog No. T27678Cas No. 959740-39-7
Alias JNJ39220675, JNJ 39220675
JNJ-39220675 (JNJ 39220675) is a selective and brain permeable histamine H3 receptor antagonist.
JNJ-39220675
🥰Excellent
Purity: 99.78%
Catalog No. T27678Alias JNJ39220675, JNJ 39220675Cas No. 959740-39-7
JNJ-39220675 (JNJ 39220675) is a selective and brain permeable histamine H3 receptor antagonist.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $293 | In Stock | |
| 5 mg | $722 | In Stock | |
| 10 mg | $987 | In Stock | |
| 25 mg | $1,520 | In Stock | |
| 50 mg | $1,980 | In Stock |
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Purity:99.78%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | JNJ-39220675 (JNJ 39220675) is a selective and brain permeable histamine H3 receptor antagonist. |
| In vivo | After establishing a reliable baseline of alcohol and water intake, systemic (subcutaneous) administration of three doses of JNJ 39220675 (0.3, 3, and 10 mg/kg) to rats in the morning (10:00 AM) significantly and dose-dependently reduced alcohol self-administration without altering saccharin self-administration in alcohol-independent rats. |
| Alias | JNJ39220675, JNJ 39220675 |
| Molecular Weight | 369.43 |
| Formula | C21H24FN3O2 |
| Cas No. | 959740-39-7 |
| Smiles | O=C(C1=CN=C(OC2=CC=C(F)C=C2)C=C1)N3CCN(CCC3)C4CCC4 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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