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Meseclazone
😃Good
Catalog No. T16353Cas No. 29053-27-8
Alias W2395, NSC297623
Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.
Meseclazone
😃Good
Catalog No. T16353Alias W2395, NSC297623Cas No. 29053-27-8
Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,520 | 6-8 weeks | |
| 50 mg | $1,980 | 6-8 weeks | |
| 100 mg | $2,500 | 6-8 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation. |
| In vivo | Intravenous administration of Meseclazone, along with other nonsteroidal anti-inflammatory drugs (NSAIDs), has been found to cause a dose-dependent reduction in bronchoconstriction. This leads to a sequence of efficacy in decreasing order as follows: isoproterenol ≈ indomethacin > fenoprofen > tolmetin > aspirin > naproxen ≈ ibuprofen > phenylbutazone > diflunisal > Meseclazone > 5-CSA. Additionally, Meseclazone demonstrates the ability to inhibit collagen-induced platelet aggregation 1 and 4 hours post oral administration[1][2]. |
| Alias | W2395, NSC297623 |
| Molecular Weight | 239.65 |
| Formula | C11H10ClNO3 |
| Cas No. | 29053-27-8 |
| Relative Density. | 1.47g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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