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Rilmakalim
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Rilmakalim
Catalog No. T26086Cas No. 132014-21-2
Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $130 | In Stock | |
| 5 mg | $320 | In Stock | |
| 10 mg | $480 | In Stock | |
| 25 mg | $786 | In Stock | |
| 50 mg | $1,080 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect. |
| In vitro | Rilmakalim (ventricular rat myocytes; patch-clamp technique) is a channel opener dose-dependently activated whole-cell currents [concentration for half-maximal activation (EC50) = 1.1 μM, Hill coefficient = 3.1, saturation concentration 10 microM].[2] |
| Molecular Weight | 401.48 |
| Formula | C21H23NO5S |
| Cas No. | 132014-21-2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 50 mg/mL (124.54 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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