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Xenin 8 acetate
🥰Excellent
Catalog No. TP2209L
Alias Xenin 8 acetate (117442-28-1 Free base)
Xenin 8 acetate is a biologically active fragment of Xenin in the neurotensin/xenopsin family. Xenin 8 acetate augments Arginine-induced insulin release (by 40%) and potentiates the glucagon responses to both Arginine (by 60%), Carbachol (by 50%).
Xenin 8 acetate
🥰Excellent
Purity: 95.54%
Catalog No. TP2209LAlias Xenin 8 acetate (117442-28-1 Free base)
Xenin 8 acetate is a biologically active fragment of Xenin in the neurotensin/xenopsin family. Xenin 8 acetate augments Arginine-induced insulin release (by 40%) and potentiates the glucagon responses to both Arginine (by 60%), Carbachol (by 50%).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $243 | In Stock | |
| 5 mg | $547 | In Stock | |
| 10 mg | $788 | In Stock | |
| 25 mg | $1,190 | In Stock | |
| 50 mg | $1,630 | In Stock | |
| 100 mg | $2,180 | In Stock |
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Purity:95.54%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Xenin 8 acetate is a biologically active fragment of Xenin in the neurotensin/xenopsin family. Xenin 8 acetate augments Arginine-induced insulin release (by 40%) and potentiates the glucagon responses to both Arginine (by 60%), Carbachol (by 50%). |
| In vitro | Xenin 8 acetate stimulates basal insulin secretion and potentiates the insulin response to glucose in a dose-dependent manner with an EC50 of 0.16 nM. Xenin 8 acetate counteracts the inhibition of glucagon release induced by increasing the glucose concentration[1]. |
| Alias | Xenin 8 acetate (117442-28-1 Free base) |
| Molecular Weight | 1106.32 |
| Formula | C53H83N15O11 |
| Smiles | CC(C[C@H](NC([C@@H](NC([C@@H](NC([C@H]1CCCN1C([C@@H](NC([C@H](CCCCN)NC([C@@H]2CCCN2C([C@@H](N)CC3=CN=CN3)=O)=O)=O)CCCNC(N)=N)=O)=O)CC4=CNC5=CC=CC=C54)=O)[C@H](CC)C)=O)C(O)=O)C.CC(O)=O |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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