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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $37 | In Stock | |
2 mg | $50 | In Stock | |
5 mg | $78 | In Stock | |
10 mg | $127 | In Stock | |
25 mg | $260 | In Stock | |
50 mg | $423 | In Stock | |
100 mg | $628 | In Stock | |
500 mg | $1,350 | In Stock | |
1 mL x 10 mM (in DMSO) | $78 | In Stock |
Description | 3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a). Displays ≥ 40-fold selectivity over other receptors: mGluR-5, mGluR-2, mGluR-4 (mGluR-4a) (IC50 > 300 μM), NMDA and GluR (AMPA) (IC50 = 250 μM). 3-MATIDA act as a neuroprotectant in cultured murine cortical cells and rat hippocampal slice cultures in vitro. |
Targets&IC50 | mGluR5:> 300 μM, mGluR1:6.3 μM, mGluR4:> 300 μM, mGluR2:> 300 μM, NMDA:250 μM, GluR(AMPA):250 μM |
Molecular Weight | 215.23 |
Formula | C8H9NO4S |
Cas No. | 518357-51-2 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 2.15 mg/mL (10 mM), Sonication is recommended. 1eq. NaOH: 50 mM | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO/1eq. NaOH
1eq. NaOH
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