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AZD-0284

Catalog No. T14369 CAS 2101291-07-8

Purity 98.00% Datasheet

AZD-0284 is an inverse agonist of the nuclear receptor RORγ. In development for the treatment of plaque psoriasis vulgaris and respiratory tract disorders[1].

AZD-0284, CAS 2101291-07-8

Pack Size	Availability	Price/USD
5 mg	inquiry	444.00
10 mg	inquiry	737.00
50 mg	inquiry	2202.00
100 mg	inquiry	3277.00
200 mg	inquiry	inquiry
500 mg	inquiry	inquiry
1 mL * 10 mM (in DMSO)	inquiry	511.00

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Purity 98.00%

Datasheet

Biological Description

Chemical Properties

Storage & Solubility Information

Description	AZD-0284 is an inverse agonist of the nuclear receptor RORγ. In development for the treatment of plaque psoriasis vulgaris and respiratory tract disorders[1].
Targets&IC50	RORγ,

Molecular Weight	524.43
Formula	C21H18F6N2O5S
CAS No.	2101291-07-8

Storage

-20℃ 3 years powder

-80℃ 2 years in solvent

Solubility Information

DMSO: 100 mg/mL (190.68 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Narjes, F, et al. The discovery of AZD0284, an inverse agonist of the nuclear receptor RORg. American Chemical Society, 2017 Drug Design and Delivery Symposium 26 October 2017

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TAK-828F Xylan Vimirogant AZD-0284 RORγt Inverse agonist 8 A-9758 S18-000003 FM26

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Answers to questions you may have can be found in the Inhibitor Handling Instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.