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Ajmaline

Catalog No. T4550 CAS 4360-12-7

Synonyms: (+)-Ajmaline, Cardiorythmine, Tachmalin, Raugalline, Tachmalin, Raugalline, Cardiorythmine, (+)-Ajmaline

Ajmaline is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.

Ajmaline, CAS 4360-12-7

Pack Size	Availability	Price/USD
5 mg	In stock	30.00
10 mg	In stock	40.00
25 mg	In stock	64.00
50 mg	In stock	99.00
100 mg	Inquiry	160.00
1 mL * 10 mM (in DMSO)	In stock	50.00

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Purity 99.67%

HNMR HPLC COA Datasheet MSDS

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Ajmaline is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.
Targets&IC50

Synonyms	(+)-Ajmaline , Cardiorythmine , Tachmalin , Raugalline , Tachmalin , Raugalline , Cardiorythmine , (+)-Ajmaline
Purity	99.67%
Molecular Weight	326.4
Formula	C20H26N2O2
CAS No.	4360-12-7

Storage

-20℃ 3 years powder

-80℃ 2 years in solvent

Solubility Information

Chloroform: Soluble

DMSO: 59 mg/mL (180.8 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Fischer F, et al. Inhibition of cardiac Kv1.5 and Kv4.3 potassium channels by the class Ia anti-arrhythmic ajmaline: mode of action.[J]. Naunyn-Schmiedeberg's Archives of Pharmacology, 2013, 386(11):991-999.

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This product is contained In the following compound libraries：

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