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Ajmaline
🥰Excellent
Catalog No. T4550Cas No. 4360-12-7
Alias Tachmalin, Raugalline, Cardiorythmine, (+)-Ajmaline
Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.
Ajmaline
🥰Excellent
Purity: 99.67%
Catalog No. T4550Alias Tachmalin, Raugalline, Cardiorythmine, (+)-AjmalineCas No. 4360-12-7
Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 100 mg | $40 | In Stock | |
| 500 mg | $92 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $29 | In Stock |
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Purity:99.67%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations. |
| Alias | Tachmalin, Raugalline, Cardiorythmine, (+)-Ajmaline |
| Molecular Weight | 326.43 |
| Formula | C20H26N2O2 |
| Cas No. | 4360-12-7 |
| Smiles | O[C@H]1C23[C@]([C@]4(N5[C@@](C2)(C1C(C4)[C@H](CC)[C@H]5O)[H])[H])(N(C)C=6C3=CC=CC6)[H] |
| Relative Density. | 1.1117 g/cm3 (Estimated) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 40 mg/mL (122.54 mM), Sonication is recommended.  Chloroform: Soluble | |||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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