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Asperuloside

Asperuloside
Asperuloside (Asperulosid) has anti-inflammatory activity.
Catalog No. T3847Cas No. 14259-45-1
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Purity:99.42%
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Asperuloside

Catalog No. T3847Cas No. 14259-45-1
Asperuloside (Asperulosid) has anti-inflammatory activity.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Pack SizePriceAvailabilityQuantity
5 mg$55In Stock
10 mg$97In Stock
25 mg$185In Stock
50 mg$276In Stock
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Product Introduction

Bioactivity
Description
Asperuloside (Asperulosid) has anti-inflammatory activity.
Kinase Assay
The chemiluminescent assay is used to confirm PCSEE MAO-A and MAO-B inhibitory effects and to test BNN and BVN hMAO-A and hMAO-B inhibition using MAO-Glo kit. Each enzyme's Arbitrary Light Unit (ALU) is measured in the presence of PCSEE, BNN, BVN, and standard DEP as an MAO-BI positive control. Briefly, hMAO-A and hMAO-B isozymes are diluted to 2× with reaction buffer (pH 7.4) and preincubated with 4× PCSEE, BNN, BVN, or DEP working solutions at RT for 30?min in white opaque 96-well plates. For determining activity inhibition, final 8.5?μg/mL concentrations of PCSEE, BNN, BVN, and DEP are used. For IC50 determination, 8× PCSEE and BNN working solutions are serially diluted using reaction buffers (pH 7.4) to make a 4× concentration. Ten points' range of PCSEE (1.0 to 250.0?μg/mL) and BNN (up to 400?μM (135.4?μg/mL)) final concentrations is used. Controls used are with and without ethanol. Ethanol solvent in controls is kept to a maximum final (volume) of ≤2%. Each isozyme is substituted with the reaction buffer for the blank. Based on our preliminary optimizations and Valley's method, the reaction is initiated by adding 4× luciferin derivative substrate (LDS) for a final (concentration) of 40 and 4?μM for hMAO-A and hMAO-B reactions, respectively. The final volume per well of each reaction is 50?μL. The reaction is optimized for the amount of A and B enzyme used to be incubated for less than 3.5?h at RT. To stop the reaction and produce the luminescence signal RLDR is added to all wells, 50?μL to each well, and incubated for a further 30?min.
AliasAsperulosid
Chemical Properties
Molecular Weight414.36
FormulaC18H22O11
Cas No.14259-45-1
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 60 mg/mL (144.8 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4134 mL12.0668 mL24.1336 mL120.6680 mL
5 mM0.4827 mL2.4134 mL4.8267 mL24.1336 mL
10 mM0.2413 mL1.2067 mL2.4134 mL12.0668 mL
20 mM0.1207 mL0.6033 mL1.2067 mL6.0334 mL
50 mM0.0483 mL0.2413 mL0.4827 mL2.4134 mL
100 mM0.0241 mL0.1207 mL0.2413 mL1.2067 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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