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CX-157
🥰Excellent
Catalog No. T15023Cas No. 205187-53-7
Alias KP 157
CX-157 (KP 157) is a novel monoamine oxidase-A (MAO-A) inhibitor for the study of depression-like neurological disorders and cancer.
CX-157
🥰Excellent
Purity: 99.35%
Catalog No. T15023Alias KP 157Cas No. 205187-53-7
CX-157 (KP 157) is a novel monoamine oxidase-A (MAO-A) inhibitor for the study of depression-like neurological disorders and cancer.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $293 | In Stock | |
| 5 mg | $722 | In Stock | |
| 10 mg | $987 | In Stock | |
| 25 mg | $1,520 | In Stock | |
| 50 mg | $1,980 | In Stock |
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Purity:99.35%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | CX-157 (KP 157) is a novel monoamine oxidase-A (MAO-A) inhibitor for the study of depression-like neurological disorders and cancer. |
| Targets&IC50 | MAO-A:（EC50）19.3 ng/ml, MAO-A:19.3 ng/ml（EC50） |
| In vivo | CX157 (60 and 80 mg) significantly inhibited the binding of [(11)C]clorgyline to brain MAO-A by 47-72% at 2 hours post-administration, with complete recovery of brain MAO-A by 24 hours post-dosing[1]. |
| Alias | KP 157 |
| Molecular Weight | 348.27 |
| Formula | C14H8F4O4S |
| Cas No. | 205187-53-7 |
| Smiles | O=S1(=O)C2=CC=C(F)C=C2OC3=CC(OCC(F)(F)F)=CC=C31 |
| Relative Density. | 1.549 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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