Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Cletoquine is a major active metabolite of Hydroxychloroquine. Cletoquine has the ability to against the chikungunya virus (CHIKV). Cletoquine has antimalarial effects and has the potential for autoimmune disease treatment.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 291.00 | |
5 mg | In stock | $ 715.00 | |
10 mg | In stock | $ 987.00 | |
25 mg | In stock | $ 1,480.00 | |
50 mg | In stock | $ 1,980.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 688.00 |
Description | Cletoquine is a major active metabolite of Hydroxychloroquine. Cletoquine has the ability to against the chikungunya virus (CHIKV). Cletoquine has antimalarial effects and has the potential for autoimmune disease treatment. |
In vivo | Hydroxychloroquine (5 mg/kg intravenously) is administered to BALB/c mice for blood and tissue to determine the content of Cletoquine. The tissue to blood concentration ratio (Kp) is ≥1, indicating the accumulation of Cletoquine in tissues. The Cletoquine Kp ratios for the various tissues are observed in the descending order of liver (114.3)>kidney (24.4)>spleen (19.3)>lungs (16.5)>heart (5.5) [3]. |
Synonyms | Desethylhydroxychloroquine |
Molecular Weight | 307.82 |
Formula | C16H22ClN3O |
CAS No. | 4298-15-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (178.68 mM)
You can also refer to dose conversion for different animals. More
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Cletoquine 4298-15-1 Microbiology/Virology Antifection Parasite Ndesethylation inhibit CHIKV P23pro-zbd antimalarial CYP2D6 Influenza Virus CYP3A4 CYP2C8 CYP3A5 Desethylhydroxychloroquine Inhibitor Hydroxychloroquine antiviral inhibitor