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Ezatiostat TFA

Catalog No. T5862
Alias TLK199, TER199(free base), Ezatiostat TFA (free base), Ezatiostat

Ezatiostat TFA (TLK199) is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity.

Ezatiostat TFA

Ezatiostat TFA

Purity: 98.74%
Catalog No. T5862Alias TLK199, TER199(free base), Ezatiostat TFA (free base), Ezatiostat
Ezatiostat TFA (TLK199) is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity.
Pack SizePriceAvailabilityQuantity
1 mg$50In Stock
5 mg$60In Stock
10 mg$102In Stock
25 mg$233In Stock
50 mg$308In Stock
100 mg$477In Stock
1 mL x 10 mM (in DMSO)$116In Stock
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Purity:98.74%
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Product Introduction

Bioactivity
Description
Ezatiostat TFA (TLK199) is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity.
In vitro
Ezatiostat is a tripeptide analog of glutathione that can selectively inhibit GSTP1-1 catalytic activity (Ki = 400 nM) with minimal effect on the related GSTα and -μ families (Kis range from 20-75 μM)[1].
AliasTLK199, TER199(free base), Ezatiostat TFA (free base), Ezatiostat
Chemical Properties
Molecular Weight643.67
FormulaC29H36F3N3O8S
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 25 mg/mL (47.2 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.5536 mL7.7680 mL15.5359 mL77.6796 mL
5 mM0.3107 mL1.5536 mL3.1072 mL15.5359 mL
10 mM0.1554 mL0.7768 mL1.5536 mL7.7680 mL
20 mM0.0777 mL0.3884 mL0.7768 mL3.8840 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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