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Fuscoside

Catalog No. T4355   CAS 131631-89-5
Synonyms: OPC 21268

Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.

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Fuscoside Chemical Structure
Fuscoside, CAS 131631-89-5
Pack Size Availability Price/USD Quantity
2 mg In stock $ 52.00
5 mg In stock $ 80.00
10 mg In stock $ 108.00
25 mg In stock $ 182.00
50 mg In stock $ 256.00
100 mg In stock $ 442.00
1 mL * 10 mM (in DMSO) In stock $ 80.00
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Purity: 99.66%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
Targets&IC50 rat V1:25 nM, human V1:8800 nM
Synonyms OPC 21268
Molecular Weight 449.54
Formula C26H31N3O4
CAS No. 131631-89-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 44.95 mg/mL (100 mM)

Ethanol: 11.24 mg/mL (25 mM)

TargetMolReferences and Literature

1. Yamamura Y,etal.PC-21268, an orally effective, nonpeptide vasopressin V1 receptor antagonist.Science. 1991 Apr 26;252(5005):572-4. 2. Imaizumi T,etal.Effects of OPC-21268, an orally effective vasopressin V1 receptor antagonist in humans.Hypertension. 1992 Jul;20(1):54-8. 3. Thibonnier M,etal.A molecular model of agonist and nonpeptide antagonist binding to the human V(1) vascular vasopressin receptor.J Pharmacol Exp Ther. 2000 Jul;294(1):195-203.

Related compound libraries

This product is contained In the following compound libraries:
Anti-Cancer Clinical Compound Library Anti-Cancer Drug Library ReFRAME Related Library Inhibitor Library Anti-Diabetic Compound Library Target-Focused Phenotypic Screening Library GPCR Compound Library Anti-Metabolism Disease Compound Library Clinical Compound Library Bioactive Compound Library

Related Products

Related compounds with same targets
Terlipressin Acetate L-371,257 Tolvaptan Desmopressin acetate (16679-58-6 free base) Conivaptan hydrochloride Dp[Tyr(methyl)2,Arg8]-Vasopressin Val9-Oxytocin Atosiban acetate

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Keywords

Fuscoside 131631-89-5 GPCR/G Protein Vasopressin Receptor OPC21268 Inhibitor OPC-21268 inhibit OPC 21268 inhibitor

 

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