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Felypressin acetate
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
Catalog No. T2568LCas No. 914453-97-7
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Purity:97.06%
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Felypressin acetate
Catalog No. T2568LCas No. 914453-97-7
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $39 | In Stock | |
| 10 mg | $64 | In Stock | |
| 25 mg | $128 | In Stock | |
| 50 mg | $197 | In Stock | |
| 100 mg | $313 | In Stock | |
| 200 mg | $468 | In Stock | |
| 500 mg | $753 | In Stock |
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Atosiban acetate
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Desmopressin acetate (16679-58-6 free base)
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T514462288-83-9
Desmopressin acetate (16679-58-6 free base) (DDAVP) is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led to its use in polyuric conditions including primary nocturnal enuresis, nocturia, and diabetes insipidus. Desmopressin acetate (16679-58-6 free base) works by limiting the amount of water that is eliminated in the urine. Desmopressin acetate (16679-58-6 free base) binds to V2 receptors in renal collecting ducts, increasing water reabsorption. It also stimulates the release of von Willebrand factor from endothelial cells by acting on the V2 receptor.
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Conopressin S acetate(111317-90-9 free base)
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Balovaptan
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Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism.
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d[Cha4]-AVP acetate(500170-27-4 free base)
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures. |
| In vitro | Felypressin is a synthetic posterior pituitary hormone with vasoconstrictive properties mediated through V1 receptors in blood vessel smooth muscle cells[4]. |
| In vivo | In Wistar rats, Felypressin (240 ng/kg; i.v.) induces a pressor effect and bradycardic effect depending on V1 receptors to induce pressor and bradycardic effects. Felypressin produces a high relationship between bradycardia and mean arterial pressure vari |
| Alias | 2-(L-Phenylalanine)-8-L-lysinevasopressin, PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond), PLV 2, PLV-2 |
| Molecular Weight | 1100.27 |
| Formula | C48H69N13O13S2 |
| Cas No. | 914453-97-7 |
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
| Solubility Information | DMSO: 10 mg/mL (9 mM), Sonication is recommended.  | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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