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LUN42518 HCl 47142-51-8(free base)

Catalog No. T8738 CAS T8738

LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.

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LUN42518 HCl 47142-51-8(free base) Chemical Structure

LUN42518 HCl 47142-51-8(free base), CAS T8738

Pack Size	Availability	Price/USD
1 mg	In stock	$ 133.00
5 mg	In stock	$ 302.00
10 mg	In stock	$ 453.00
25 mg	In stock	$ 747.00
50 mg	In stock	$ 1,050.00
100 mg	In stock	$ 1,420.00
1 mL * 10 mM (in DMSO)	In stock	$ 298.00

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Purity: 99.85%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.

Molecular Weight	317.81
Formula	C17H20ClN3O
CAS No.	T8738

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 22.5 mg/mL (70.8 mM)

References and Literature

1. J.A. Parihar, et al. Alkylation of diphenylamines with chloroacetonitrile: a new entry to phentolamine analogues. Journal of Chemical Research (2004), (3), 220-222.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Anti-Neurodegenerative Disease Compound Library GPCR Compound Library Membrane Protein-targeted Compound Library Neuronal Signaling Compound Library Anti-Cardiovascular Disease Compound Library NO PAINS Compound Library Anti-Cancer Compound Library Anti-Alzheimer's Disease Compound Library Neurotransmitter Receptor Compound Library

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Related compounds with same targets

Tienoxolol FA Deriglidole Betaxolol hydrochloride Salmeterol Xinafoate Dipivefrin hydrochloride Efloxate Indacaterol maleate Ancarolol

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

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