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Multi-kinase inhibitor 1

Catalog No. T4191 CAS 778274-97-8

Synonyms: Platelet-derived growth factor receptor, inhibit, Bcr-Abl, SCFR, CD117, Multi-kinase inhibitor 1, Multi-kinase inhibitor I, c-Kit, Multi kinase inhibitor 1, PDGFR, Multikinase inhibitor 1, Inhibitor

Multi-kinase inhibitor I is a Multi-kinase inhibitor.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Multi-kinase inhibitor 1, CAS 778274-97-8

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Multi-kinase inhibitor I is a Multi-kinase inhibitor.

Synonyms	Platelet-derived growth factor receptor, inhibit, Bcr-Abl, SCFR, CD117, Multi-kinase inhibitor 1, Multi-kinase inhibitor I, c-Kit, Multi kinase inhibitor 1, PDGFR, Multikinase inhibitor 1, Inhibitor
Molecular Weight	418.376
Formula	C20H17F3N4O3
CAS No.	778274-97-8

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Chang Hsu Y, et al. Discovery of BPR1K871, a quinazoline based, multi-kinase inhibitor for the treatment of AML and solid tumors: Rational design, synthesis, in vitro and in vivo evaluation. Oncotarget. 2016 Nov 15 2. García-Vilas JA, et al. The noni anthraquinone damnacanthal is a multi-kinase inhibitor with potent anti-angiogenic effects. Cancer Lett. 2017 Jan 28;385:1-11 3. Li Y, et al. The molecular mechanisms of a novel multi-kinase inhibitor ZLJ33 in suppressing pancreatic cancer growth. Cancer Lett. 2015 Jan 28;356(2 Pt B):392-403

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Fluorochemical Library Kinase Inhibitor Library Bioactive Compound Library

Related Products

Related compounds with same targets

CZC-8004 Sabutoclax BGG463 Nilotinib hydrochloride Dasatinib hydrochloride Pivanex Cenisertib SIAIS178

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.