Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Pimelic diphenylamide 106 (RGFA-8) is a slow, tight-binding inhibitor of class I HDAC (with IC50 values of 150 nM , 760 nM and 370 nM for HDAC 1, 2, and 3, respectively), showing no activity against class II HDACs.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 42.00 | |
10 mg | In stock | $ 67.00 | |
25 mg | In stock | $ 115.00 | |
50 mg | In stock | $ 197.00 | |
100 mg | In stock | $ 359.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 46.00 |
Description | Pimelic diphenylamide 106 (RGFA-8) is a slow, tight-binding inhibitor of class I HDAC (with IC50 values of 150 nM , 760 nM and 370 nM for HDAC 1, 2, and 3, respectively), showing no activity against class II HDACs. |
Targets&IC50 | HDAC 3:370 nM, HDAC2:760 nM, HDAC 1:150 nM |
Synonyms | Histone Deacetylase Inhibitor VII, TC-H 106, RGFA-8 |
Molecular Weight | 339.43 |
Formula | C20H25N3O2 |
CAS No. | 937039-45-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (162.04 mM)
You can also refer to dose conversion for different animals. More
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Pimelic diphenylamide 106 937039-45-7 Chromatin/Epigenetic DNA Damage/DNA Repair HDAC Pimelic Diphenylamide-106 TC-H106 Pimelic Diphenylamide106 Histone Deacetylase Inhibitor VII Inhibitor TC-H-106 RGFA8 TC-H 106 inhibit RGFA-8 Histone deacetylases RGFA 8 inhibitor