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Asenapine hydrochloride
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Catalog No. T22589Cas No. 1261398-77-9
Alias Org 5222 hydrochloride
Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder.
Asenapine hydrochloride
😃Good
Catalog No. T22589Alias Org 5222 hydrochlorideCas No. 1261398-77-9
Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $69 | 7-10 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder. |
| Targets&IC50 | D2 receptor:1.3 nM (Ki), 5-HT2C receptor:0.03 nM (Ki), D3 receptor:0.42 nM (Ki), 5-HT2A receptor:0.06 nM (Ki), D4 receptor:1.1 nM (Ki), 5-HT7 receptor:0.13 nM (Ki), sPLA2:2.5 nM (Ki) |
| In vitro | Asenapine hydrochloride acts as an antagonist of 5-HT2A receptors and D2 receptors, commonly used in research related to neurological disorders[2]. |
| Alias | Org 5222 hydrochloride |
| Molecular Weight | 322.23 |
| Formula | C17H17Cl2NO |
| Cas No. | 1261398-77-9 |
| Smiles | Cl.[H][C@]12CN(C)C[C@]1([H])c1cc(Cl)ccc1Oc1ccccc21 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||
| Solubility Information | DMSO: 1 mg/mL (3.10 mM), Sonication is recommended. | ||||||||||
Solution Preparation Table | |||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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